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  • Faculty of Pharmacy
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  • The Role of Metabolism in Drug Design
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Course Title Code Compulsory/Elective Laboratory + Practice ECTS
The Role of Metabolism in Drug Design ECZ898 X. SEMESTER 1+0 1.5
Language of Instruction Türkçe
Course Type Uzmanlık Alanı Dersleri
Course Instructor(s) DOÇ. DR. DERYA OSMANİYE
Mode of Delivery Face to face learning.
Prerequisites There is no prerequisite or co-requisite for this course.
Courses Recomended
Recommended Reading List
Assessment methods and criteria 1 Mid Term Exam, 1 Final Exam
Work Placement None.
Catalog Content Introduction to Drug Metabolism; Phase I Reactions; Phase II Reactions; Drug Structure and Metabolism; Effect of Stereochemical Factors on Metabolism; Pharmacokinetic Relationship with Metabolization through Prodrug Definition; Drug Design for Reducing Toxicity by Examining Probable Toxic Metabolites of Drugs; Effect of Metabolization on Bioavailability; Effect of Metabolism on Drug Activity; Active Metabolite Approach in Drug Design; The Role of Metabolism in New Drug Development.

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