Anadolu Info Package Anadolu Info Package
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General Information Departments Educational Staff Administration Contact
  • Faculty of Pharmacy
  • Course Structure Diagram with Credits
  • Computer-Aided Drug Design
  • Content
  • Description
  • Content
  • Learning Outcomes
  • Learning Activities and Teaching Methods
  • Course's Contribution to Prog.
  • Assessment Methods

Weeks Topics
Week - 1 Computer methods in the Pharmaceutical and Medicinal Chemistry, it’s importance on drug design,
Week - 2 Computer methods in the Pharmaceutical and Medicinal Chemistry, it’s importance on drug design,
Week - 3 ligand-based drug design: Traditional 2D QSAR, Pharmacophor Analyses,
Week - 4 3D QSAR ((CoMFA (Comparative Molecular Field Analysis), CoMSIA (Comparative Molecular Similarity Indices Analysis ) Methods),
Week - 5 3D QSAR ((CoMFA (Comparative Molecular Field Analysis), CoMSIA (Comparative Molecular Similarity Indices Analysis ) Methods),
Week - 6 4D, 5D and 6D-QSAR; (structural-based drug design),
Week - 7 (structural-based drug design), Molecular modelling,
Week - 8 (structural-based drug design), Molecular modelling,
Week - 9 Docking and imaging, molecular mechanics and molecular dinamic methods,
Week - 10 virtual screening, pharmacological modelling,
Week - 11 virtual screening, pharmacological modelling,
Week - 12 Library design, High-throughput screening (HTS),
Week - 13 de novo (synthetic) drug design,
Week - 14 Computer-aided design of enzyme inhibitors as drug-targets.

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